Synthesis and Biological Activities of Thio-avarol Derivatives
Abstract
Eleven new thio-avarol derivatives (3-13) were synthesized. Their antimicrobial, brine shrimp lethality, and free-radical scavenging activities and acetylcholinesterase inhibition, together with 12 already reported semisynthetic thioavarol derivatives (14-25), were evaluated. Structure-activity relationships among these thio derivatives were determined.
Source:
Journal of Natural Products, 2008, 71, 11, 1850-1853Publisher:
- Amer Chemical Soc, Washington
Funding / projects:
- CNR-RomeConsiglio Nazionale delle Ricerche (CNR)
- Italian Minister of Foreign Affairs fellowship
DOI: 10.1021/np800318m
ISSN: 0163-3864
PubMed: 19007183
WoS: 000261335800011
Scopus: 2-s2.0-58149168976
Collections
Institution/Community
Institut za multidisciplinarna istraživanjaTY - JOUR AU - Pejin, Boris AU - Iodice, Carmine AU - Tommonaro, Giuseppina AU - De Rosa, Salvatore PY - 2008 UR - http://rimsi.imsi.bg.ac.rs/handle/123456789/281 AB - Eleven new thio-avarol derivatives (3-13) were synthesized. Their antimicrobial, brine shrimp lethality, and free-radical scavenging activities and acetylcholinesterase inhibition, together with 12 already reported semisynthetic thioavarol derivatives (14-25), were evaluated. Structure-activity relationships among these thio derivatives were determined. PB - Amer Chemical Soc, Washington T2 - Journal of Natural Products T1 - Synthesis and Biological Activities of Thio-avarol Derivatives EP - 1853 IS - 11 SP - 1850 VL - 71 DO - 10.1021/np800318m ER -
@article{ author = "Pejin, Boris and Iodice, Carmine and Tommonaro, Giuseppina and De Rosa, Salvatore", year = "2008", abstract = "Eleven new thio-avarol derivatives (3-13) were synthesized. Their antimicrobial, brine shrimp lethality, and free-radical scavenging activities and acetylcholinesterase inhibition, together with 12 already reported semisynthetic thioavarol derivatives (14-25), were evaluated. Structure-activity relationships among these thio derivatives were determined.", publisher = "Amer Chemical Soc, Washington", journal = "Journal of Natural Products", title = "Synthesis and Biological Activities of Thio-avarol Derivatives", pages = "1853-1850", number = "11", volume = "71", doi = "10.1021/np800318m" }
Pejin, B., Iodice, C., Tommonaro, G.,& De Rosa, S.. (2008). Synthesis and Biological Activities of Thio-avarol Derivatives. in Journal of Natural Products Amer Chemical Soc, Washington., 71(11), 1850-1853. https://doi.org/10.1021/np800318m
Pejin B, Iodice C, Tommonaro G, De Rosa S. Synthesis and Biological Activities of Thio-avarol Derivatives. in Journal of Natural Products. 2008;71(11):1850-1853. doi:10.1021/np800318m .
Pejin, Boris, Iodice, Carmine, Tommonaro, Giuseppina, De Rosa, Salvatore, "Synthesis and Biological Activities of Thio-avarol Derivatives" in Journal of Natural Products, 71, no. 11 (2008):1850-1853, https://doi.org/10.1021/np800318m . .